Volume 107

European Journal of Medicinal Chemistry

Volume 107

1

Design of α7 nicotinic acetylcholine receptor ligands using the (het)Aryl-1,2,3-triazole core: Synthesis, in vitro evaluation and SAR studies

Ouach, Aziz, Pin, Frederic, Bertrand, Emilie, Vercouillie, Johnny, Gulhan, Zuhal, Mothes, Céline, Deloye, Jean-Bernard, Guilloteau, Denis, Suzenet, Franck, Chalon, Sylvie, Routier, Sylvain

Journal:

European Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 1.75 MB

english, 2016

2

Synthesis and in vitro antitumor evaluation of dihydroartemisinin-cinnamic acid ester derivatives

Xu, Cang-Cang, Deng, Ting, Fan, Meng-Lin, Lv, Wen-Bo, Liu, Ji-Hua, Yu, Bo-Yang

Journal:

European Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 1.58 MB

english, 2016

3

Novel nonsecosteroidal VDR ligands with phenyl-pyrrolyl pentane skeleton for cancer therapy

Ge, Zhixin, Hao, Meixi, Xu, Meng, Su, Zhigui, Kang, Zisheng, Xue, Lingjing, Zhang, Can

Journal:

European Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 1.43 MB

english, 2016

4

Design and synthesis of a C7-aryl piperlongumine derivative with potent antimicrotubule and mutant p53-reactivating properties

Punganuru, Surendra R., Madala, Hanumantha Rao, Venugopal, Sanjay N., Samala, Ramakrishna, Mikelis, Constantinos, Srivenugopal, Kalkunte S.

Journal:

European Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 1.60 MB

english, 2016

5

The biphosphinic paladacycle complex induces melanoma cell death through lysosomal–mitochondrial axis modulation and impaired autophagy

Gigli, Rafael, Pereira, Gustavo J.S., Antunes, Fernanda, Bechara, Alexandre, Garcia, Daniel M., Spindola, Daniel G., Jasiulionis, Mirian G., Caires, Antonio C.F., Smaili, Soraya S., Bincoletto, Claudi

Journal:

European Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 2.26 MB

english, 2016

6

Comparative study of structural models of Leishmania donovani and human GDP-mannose pyrophosphorylases

Daligaux, Pierre, Bernadat, Guillaume, Tran, Linh, Cavé, Christian, Loiseau, Philippe M., Pomel, Sébastien, Ha-Duong, Tâp

Journal:

European Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 4.60 MB

english, 2016

7

Extended structure–activity study of thienopyrimidine-based EGFR inhibitors with evaluation of drug-like properties

Bugge, Steffen, Buene, Audun Formo, Jurisch-Yaksi, Nathalie, Moen, Ingri Ullestad, Skjønsfjell, Ellen Martine, Sundby, Eirik, Hoff, Bård Helge

Journal:

European Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 2.31 MB

english, 2016

8

Anticonvulsant activity, crystal structures, and preliminary safety evaluation of N-trans-cinnamoyl derivatives of selected (un)modified aminoalkanols

Gunia-Krzyżak, Agnieszka, Żesławska, Ewa, Słoczyńska, Karolina, Koczurkiewicz, Paulina, Nitek, Wojciech, Żelaszczyk, Dorota, Szkaradek, Natalia, Waszkielewicz, Anna M., Pękala, Elżbieta, Marona, Henry

Journal:

European Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 1.32 MB

english, 2016

9

Design, synthesis, and biological evaluation of novel quinazolinyl-diaryl urea derivatives as potential anticancer agents

Chen, Jia-Nian, Wang, Xian-Fu, Li, Ting, Wu, De-Wen, Fu, Xiao-Bo, Zhang, Guang-Ji, Shen, Xing-Can, Wang, Heng-Shan

Journal:

European Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 2.48 MB

english, 2016

10

Anti-Candida activity and cytotoxicity of a large library of new N-substituted-1,3-thiazolidin-4-one derivatives

De Monte, Celeste, Carradori, Simone, Bizzarri, Bruna, Bolasco, Adriana, Caprara, Federica, Mollica, Adriano, Rivanera, Daniela, Mari, Emanuela, Zicari, Alessandra, Akdemir, Atilla, Secci, Daniela

Journal:

European Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 2.43 MB

english, 2016

11

Discovery of a marine-derived bis-indole alkaloid fascaplysin, as a new class of potent P-glycoprotein inducer and establishment of its structure–activity relationship

Manda, Sudhakar, Sharma, Sadhana, Wani, Abubakar, Joshi, Prashant, Kumar, Vikas, Guru, Santosh K., Bharate, Sonali S., Bhushan, Shashi, Vishwakarma, Ram A., Kumar, Ajay, Bharate, Sandip B.

Journal:

European Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 829 KB

english, 2016

12

Potent and selective N-(4-sulfamoylphenyl)thiourea-based GPR55 agonists

Yrjölä, Sari, Parkkari, Teija, Navia-Paldanius, Dina, Laitinen, Tuomo, Kaczor, Agnieszka A., Kokkola, Tarja, Adusei-Mensah, Frank, Savinainen, Juha R., Laitinen, Jarmo T., Poso, Antti, Alexander, Amy,

Journal:

European Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 2.54 MB

english, 2016

13

Hybrid triazoles: Design and synthesis as potential dual inhibitor of growth and efflux inhibition in tuberculosis

Dixit, Prasad P., Dixit, Prashant P., Thore, Shivajirao N.

Journal:

European Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 399 KB

english, 2016

14

3-(Dipropylamino)-5-hydroxybenzofuro[2,3-f]quinazolin-1(2H)-one (DPA-HBFQ-1) plays an inhibitory role on breast cancer cell growth and progression

Rizza, Pietro, Pellegrino, Michele, Caruso, Anna, Iacopetta, Domenico, Sinicropi, Maria Stefania, Rault, Sylvain, Lancelot, Jean Charles, El-Kashef, Hussein, Lesnard, Aurelien, Rochais, Christophe, Da

Journal:

European Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 1.51 MB

english, 2016

15

Structure–activity relationship study of anticancer thymidine–quinoxaline conjugates under the low radiance of long wavelength ultraviolet light for photodynamic therapy

Zhang, Dejun, Liu, Huaming, Wei, Qiong, Zhou, Qibing

Journal:

European Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 2.05 MB

english, 2016

16

New highly active antiplatelet agents with dual specificity for platelet P2Y1 and P2Y12 adenosine diphosphate receptors

Yanachkov, Ivan B., Chang, Hung, Yanachkova, Milka I., Dix, Edward J., Berny-Lang, Michelle A., Gremmel, Thomas, Michelson, Alan D., Wright, George E., Frelinger, Andrew L.

Journal:

European Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 1.12 MB

english, 2016

17

Editorial board

Journal:

European Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 48 KB

english, 2016

18

Graphical contents list

Journal:

European Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 1.27 MB

english, 2016

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