Volume 58; Issue 9

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Il Farmaco
Volume 58; Issue 9

Il Farmaco

Volume 58; Issue 9

1

Ibuprofen quality control by electrochromatography

M.G Quaglia, E Donati, S Fanali, P Catarcini

Journal:

Year:

2003

Language:

english

File:

PDF, 241 KB

english, 2003

2

Photostability studies on the furosemide–triamterene drug association

J Fiori, R Ballardini, V Andrisano, V Cavrini

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Year:

2003

Language:

english

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PDF, 252 KB

english, 2003

3

3D QSAR studies for the β-tubulin binding site of microtubule-stabilizing anticancer agents (MSAAs): A pseudoreceptor model for taxanes based on the experimental structure of tubulin

Laura Maccari, Fabrizio Manetti, Federico Corelli, Maurizio Botta

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Year:

2003

Language:

english

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PDF, 323 KB

english, 2003

4

Synthesis and antagonistic activity at muscarinic receptor subtypes of some derivatives of diphenidol

Lucilla Varoli, Piero Angeli, Michela Buccioni, Silvia Burnelli, Andrea Cavalli, Gabriella Marucci, Maurizio Recanatini

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Year:

2003

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english

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PDF, 238 KB

english, 2003

5

Quinoxaline chemistry. Part 16. 4-Substituted anilino and 4-substituted phenoxymethyl pyrrolo[1,2-a]quinoxalines and N-[4-(pyrrolo[1,2-a]quinoxalin-4-yl)amino and hydroxymethyl]benzoyl glutamates. Synthesis and evaluation of in vitro biological activity

Sergio Alleca, Paola Corona, Mario Loriga, Giuseppe Paglietti, Roberta Loddo, Valeria Mascia, Bernardetta Busonera, Paolo La Colla

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Year:

2003

Language:

english

File:

PDF, 298 KB

english, 2003

6

Synthesis and affinity for serotonin and dopamine transporters of some benzophenone oxime ether derivatives

Annalina Lapucci, Susanna Nencetti, Gian Carlo Demontis

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Year:

2003

Language:

english

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PDF, 186 KB

english, 2003

7

Synthesis and antimycobacterial activity of (3,4-diaryl-3H-thiazol-2-ylidene)-hydrazide derivatives

Maria Grazia Mamolo, Valeria Falagiani, Daniele Zampieri, Luciano Vio, Elena Banfi, Giuditta Scialino

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Year:

2003

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english

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PDF, 215 KB

english, 2003

8

N-Homolupinanoyl and N-(ω-lupinylthio)alkanoyl derivatives of some tricyclic systems as ligands for muscarinic M1 and M2 receptor subtypes

Bruno Tasso, Anna Sparatore, Fabio Sparatore

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Year:

2003

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english

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PDF, 245 KB

english, 2003

9

Comparative QSAR of the sulfonamide function

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Year:

2003

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english

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PDF, 193 KB

english, 2003

10

Synthesis and vasodilating properties of N-alkylamide derivatives of 4-amino-3-furoxancarboxylic acid and related azo derivatives

I.V Ovchinnikov, A.S Kulikov, N.N Makhova, P Tosco, A Di Stilo, R Fruttero, A Gasco

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Year:

2003

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english

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PDF, 194 KB

english, 2003

11

Synthesis and biological evaluation of new amino acids structurally related to the antitumor agent acivicin

Paola Conti, Gabriella Roda, Helena Stabile, Maria Antonietta Vanoni, Bruno Curti, Marco De Amici

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Year:

2003

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english

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PDF, 265 KB

english, 2003

12

Docking experiments showing similar recognition patterns of paclitaxel when interacting with different macromolecular targets

Stefano Alcaro, Danilo Battaglia, Francesco Ortuso

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Year:

2003

Language:

english

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PDF, 519 KB

english, 2003

13

Effects of leflunomide on human cartilage

Annamaria Panico, Venera Cardile, Barbara Gentile, Floriana Garufi, Paolo Fama', Giuseppe Bonfiglio, Giuseppe Ronsisvalle

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Year:

2003

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english

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PDF, 244 KB

english, 2003

14

Synthesis and prostaglandin synthase inhibitory activity of new aromatic O-alkyloxime ethers substituted with methylsulfonamido or methylsulfonyl groups on their aliphatic portion

Aldo Balsamo, Francesca Mancini, Claudio Milanese, Elisabetta Orlandini, Gabriella Ortore, Mario Pinza, Simona Rapposelli, Armando Rossello

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Year:

2003

Language:

english

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PDF, 320 KB

english, 2003

15

2-Pyrrolidinone moiety is not critical for the cognition-enhancing activity of piracetam-like drugs

Serena Scapecchi, Cecilia Martelli, Carla Ghelardini, Luca Guandalini, Elisabetta Martini, Fulvio Gualtieri

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Year:

2003

Language:

english

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PDF, 310 KB

english, 2003

16

Synthesis and in vitro pharmacology of novel heterocyclic muscarinic ligands

Marco De Amici, Paola Conti, Ezio Fasoli, Elisabetta Barocelli, Vigilio Ballabeni, Simona Bertoni, Mariannina Impicciatore, Bryan L Roth, Paul Ernsberger, Carlo De Micheli

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Year:

2003

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english

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PDF, 284 KB

english, 2003

17

Chromophore-modified bis-benzo[g]indole carboxamides: synthesis and antiproliferative activity of bis-benzo[g]indazole-3-carboxamides and related dimers

Gérard A Pinna, Maria A Pirisi, Jean-Mario Mussinu, Gabriele Murineddu, Giovanni Loriga, Amedeo Pau, Giuseppe E Grella

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Year:

2003

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english

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PDF, 356 KB

english, 2003

18

Synthesis of N-substituted-N-acylthioureas of 4-substituted piperazines endowed with local anaesthetic, antihyperlipidemic, antiproliferative activities and antiarrythmic, analgesic, antiaggregating actions

Angelo Ranise, Andrea Spallarossa, Olga Bruno, Silvia Schenone, Paola Fossa, Giulia Menozzi, Francesco Bondavalli, Luisa Mosti, Annalisa Capuano, Filomena Mazzeo, Giuseppe Falcone, Walter Filippelli

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Year:

2003

Language:

english

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PDF, 514 KB

english, 2003

19

Isolation and pharmacological activities of the Tecoma stans alkaloids

Luca Costantino, Laura Raimondi, Renato Pirisino, Tiziana Brunetti, Pompeo Pessotto, Fabio Giannessi, Arlete Paulino Lins, Daniela Barlocco, Luciano Antolini, Samia A El-Abady

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Year:

2003

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english

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PDF, 226 KB

english, 2003

20

1,2-Dithiolan-3-ones and derivatives structurally related to leinamycin. Synthesis and biological evaluation

Raul Salvetti, Giovanni Martinetti, Daniela Ubiali, Massimo Pregnolato, Giuseppe Pagani

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Year:

2003

Language:

english

File:

PDF, 195 KB

english, 2003

21

Synthesis and activity of novel glutathione analogues containing an urethane backbone linkage

I Cacciatore, A.M Caccuri, A Di Stefano, G Luisi, M Nalli, F Pinnen, G Ricci, P Sozio

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Year:

2003

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english

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PDF, 247 KB

english, 2003

22

4-Substituted 1,5-diarylpyrazole, analogues of celecoxib: synthesis and preliminary evaluation of biological properties

Giulia Menozzi, Luisa Merello, Paola Fossa, Luisa Mosti, Antonietta Piana, Francesca Mattioli

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Year:

2003

Language:

english

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PDF, 392 KB

english, 2003

23

Preliminary biological assay on cerebroside mixture from Euphorbia nicaeensis All. Isolation and structure determination of five glucocerebrosides

F. Cateni, J. Zilic, G. Falsone, F. Hollan, F. Frausin, V. Scarcia

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Year:

2003

Language:

english

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PDF, 278 KB

english, 2003

24

In vitro anti-acanthamoeba action by thioureidic derivatives

Carmela Saturnino, Mariafrancesca Buonerba, Nicola Paesano, Jean-Charles Lancelot, Giovanni De Martino

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Year:

2003

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english

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PDF, 188 KB

english, 2003

25

Antioxidant activity of thioureidic derivatives I

Carmela Saturnino, Marta D'Auria, Nicola Paesano, Daniele Saponiero, Giuseppina Cioffi, Mariafrancesca Buonerba, Giovanni De Martino

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Year:

2003

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english

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PDF, 213 KB

english, 2003

26

Enzyme activities of tryptophan metabolism along the kynurenine pathway in various species of animals

Graziella Allegri, Carlo V.L Costa, Antonella Bertazzo, Monica Biasiolo, Eugenio Ragazzi

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Year:

2003

Language:

english

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PDF, 249 KB

english, 2003

27

Determination of a novel angiotensin-AT1 antagonist CR 3210 in biological samples by HPLC

M. Rizzo, M. Anzini, A. Cappelli, S. Vomero, D. Ventrice, G. De Sarro, S. Procopio, N. Costa, F. Makovec

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Year:

2003

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english

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PDF, 232 KB

english, 2003

28

2-Aryl-3-phenylamino-4,5-dihydro-2h-benz[g]indazoles with analgesic activity

Silvia Schenone, Olga Bruno, Angelo Ranise, Chiara Brullo, Francesco Bondavalli, Walter Filippelli, Filomena Mazzeo, Annalisa Capuano, Giuseppe Falcone

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Year:

2003

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english

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PDF, 188 KB

english, 2003

29

Towards new neuroprotective agents: design and synthesis of 4H-thieno[2,3-c] isoquinolin-5-one derivatives as potent PARP-1 inhibitors

Roberto Pellicciari, Emidio Camaioni, Gabriele Costantino, Maura Marinozzi, Antonio Macchiarulo, Flavio Moroni, Benedetto Natalini

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Year:

2003

Language:

english

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PDF, 484 KB

english, 2003

30

Synthesis of 3- or 4-phenyl-1,8-naphthyridine derivatives and evaluation of antimycobacterial and antimicrobial activity

Muwaffag Badawneh, Laura Bellini, Tiziana Cavallini, Jalal Al jamal, Clementina Manera, Giuseppe Saccomanni, Pier Luigi Ferrarini

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Year:

2003

Language:

english

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PDF, 228 KB

english, 2003

31

Synthesis, X-ray crystal structure and biological properties of acetylenic flavone derivatives

Roberto Artali, Pier Luigi Barili, Gabriella Bombieri, Paolo Da Re, Nicoletta Marchini, Fiorella Meneghetti, Piero Valenti

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Year:

2003

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english

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PDF, 376 KB

english, 2003

32

Structural characterization of a dipeptide compound with immunostimulant activity: 3-(5-thioxo-l-prolyl)-l-thiazolidine-4-carboxylic acid

R Artali, G Bombieri, F Meneghetti, D Nava, E Ragg, R Stradi

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Year:

2003

Language:

english

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PDF, 319 KB

english, 2003

33

The role of HB-donor groups in the heterocyclic polar fragment of H3-antagonists.: I. Synthesis and biological assays

Valentina Zuliani, Fabrizio Bordi, Mirko Rivara, Claudia Silva, Federica Vacondio, Giovanni Morini, Silvia Rivara, Elisabetta Barocelli, Vigilio Ballabeni, Simona Bertoni, Francesca Magnanini, Pier Vi

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Year:

2003

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english

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PDF, 279 KB

english, 2003

34

Inhibition of drug binding to human serum albumin by cholecystographic agents

Carlo Bertucci, Samanta Cimitan

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Year:

2003

Language:

english

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PDF, 659 KB

english, 2003

35

Multivariate least squares regression applied to the spectrophotometric analysis of manidipine and its main photoproduct

Gaetano Ragno, Francesca Aiello, Antonio Garofalo, Giuseppina Ioele, Maria Stefania Sinicropi

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Year:

2003

Language:

english

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PDF, 219 KB

english, 2003

36

Design, synthesis and biological evaluation of ambenonium derivatives as AChE inhibitors

Maria Laura Bolognesi, Andrea Cavalli, Vincenza Andrisano, Manuela Bartolini, Rita Banzi, Alessandra Antonello, Michela Rosini, Carlo Melchiorre

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Year:

2003

Language:

english

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PDF, 367 KB

english, 2003

37

Congo red analogues as potential anti-prion agents

Stefania Villa, Giorgio Cignarella, Daniela Barlocco, Marco Gervasoni, Gabriella Carcassola, Laura Giannino, Paolo Mantegazza

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Year:

2003

Language:

english

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PDF, 306 KB

english, 2003

38

Synthesis and pharmacological evaluation of new N-methyl-arylpyrrolidinols with analgesic activity

Simona Collina, Ornella Azzolina, Dina Vercesi, Gloria Brusotti, Daniela Rossi, Annalisa Barbieri, Enrica Lanza, Laura Mennuni, Stefano Alcaro, Danilo Battaglia, Laura Linati, Victor Ghislandi

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Year:

2003

Language:

english

File:

PDF, 446 KB

english, 2003

39

Validation of a GC/MS method for the determination of tramadol in human plasma after intravenous bolus

Veniero Gambaro, Claudio Benvenuti, Lucia De Ferrari, Lucia Dell'Acqua, Fiorenza Farè

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Year:

2003

Language:

english

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PDF, 189 KB

english, 2003

40

An investigation of the biological effect of structural modifications of isothiosemicarbazones and their cyclic analogues

E Maccioni, M.C Cardia, S Distinto, L Bonsignore, A De Logu

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Year:

2003

Language:

english

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PDF, 234 KB

english, 2003

41

2-(Dialkylamino)-4H-1-benzopyran-4-one derivatives modify chloride conductance in CFTR expressing cells

Mauro Mazzei, Erika Nieddu, Chiara Folli, Emanuela Caci, Louis V.J Galietta

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Year:

2003

Language:

english

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PDF, 482 KB

english, 2003

42

pH-Partition profiles of 4-(3-oxo-1,2-benzisothiazolin-2-yl)phenyl and phenoxyalkanoic acids

Claudia Silva, Marco Mor, Federica Vacondio, Valentina Zuliani, Pier Vincenzo Plazzi

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Year:

2003

Language:

english

File:

PDF, 218 KB

english, 2003

43

Benzoazepine derivative as potent antagonists of the glycine binding site associated to the NMDA receptor

Romano Di Fabio, Fabrizio Micheli, Davide Baraldi, Barbara Bertani, Nadia Conti, Giovanna Dal Forno, Aldo Feriani, Daniele Donati, Carla Marchioro, Tommaso Messeri, Andrea Missio, Alessandra Pasquarel

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Year:

2003

Language:

english

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PDF, 403 KB

english, 2003

44

A study on the release mechanism of drugs from hydrophilic partially coated perforated matrices

Maria Edvige Sangalli, Alessandra Maroni, Lucia Zema, Matteo Cerea, Ubaldo Conte, Andrea Gazzaniga

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Year:

2003

Language:

english

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PDF, 263 KB

english, 2003

45

QSAR and the role of luck in research

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2003

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english

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PDF, 147 KB

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46

Foreword

Roberto Pellicciari

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Year:

2003

Language:

english

File:

PDF, 124 KB

english, 2003