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1H-Imidazo[4,5-c]pyridine-4-carbonitrile as cathepsin S inhibitors: Separation of desired cellular activity from undesired tissue accumulation through optimization of basic nitrogen pka
Wullie Arbuckle, Mark Baugh, Simone Belshaw, D. Jonathan Bennett, John Bruin, Jiaqiang Cai, Kenneth S. Cameron, Chris Claxton, Maureen Dempster, Kathryn Everett, Xavier Fradera, William Hamilton, PhilVolume:
21
Year:
2011
Language:
english
Pages:
4
DOI:
10.1016/j.bmcl.2010.12.065
File:
PDF, 363 KB
english, 2011