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Discovery of Biaryl Amides as Potent, Orally Bioavailable, and CNS Penetrant RORγt Inhibitors
Wang, Yonghui, Cai, Wei, Cheng, Yaobang, Yang, Ting, Liu, Qian, Zhang, Guifeng, Meng, Qinghua, Han, Fangbin, Huang, Yafei, Zhou, Ling, Xiang, Zhijun, Zhao, Yong-Gang, Xu, Yan, Cheng, Ziqiang, Lu, SijiVolume:
6
Language:
english
Journal:
ACS Medicinal Chemistry Letters
DOI:
10.1021/acsmedchemlett.5b00122
Date:
July, 2015
File:
PDF, 544 KB
english, 2015