Volume 12; Issue 24

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Bioorganic & Medicinal Chemistry Letters
Volume 12; Issue 24

Bioorganic & Medicinal Chemistry Letters

Volume 12; Issue 24

1

Unique hole-Trapping property of the degenerate base,2-amino-7-deazaadenine

Akimitsu Okamoto, Kazuo Tanaka, Isao Saito

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 171 KB

english, 2002

2

Characterization of mono- and diaminopyrimidine derivatives as novel, nonpeptide gonadotropin releasing hormone (GnRH) receptor antagonists

David R Luthin, Yufeng Hong, Eileen Tompkins, Kenna L Anderes, Genevieve Paderes, Eugenia A Kraynov, Mary A Castro, Karen D Nared-Hood, Rosemary Castillo, Margaret Gregory, Haresh Vazir, John M May, M

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 176 KB

english, 2002

3

An expedient synthesis of Nα-protected-l-tetrahydrofuranylglycine and its application in the synthesis of novel substrate based inhibitors of HIV-1 protease

S. Rajesh, Ei'ichi Ami, Tomoya Kotake, Tooru Kimura, Yoshio Hayashi, Yoshiaki Kiso

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 125 KB

english, 2002

4

Reductively activated disulfide prodrugs of paclitaxel

Vivekananda M. Vrudhula, John F. MacMaster, Zhengong Li, David E. Kerr, Peter D. Senter

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 146 KB

english, 2002

5

Novel 1′,1′-chain substituted Δ8-tetrahydrocannabinols

Demetris P. Papahatjis, Spyros P. Nikas, Thanos Andreou, Alexandros Makriyannis

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 131 KB

english, 2002

6

Synthesis, radiolabeling and preliminary biological evaluation of radiolabeled 5-methyl-6-nitroquipazine, a potential radioligand for the serotonin transporter

Johan Sandell, Meixiang Yu, Patrick Emond, Lucette Garreau, Sylvie Chalon, Kjell Någren, Denis Guilloteau, Christer Halldin

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 119 KB

english, 2002

7

Antitrypanosomal activities and cytotoxicity of 5-nitro-2-furancarbohydrazides

Régis Millet, Louis Maes, Valérie Landry, Christian Sergheraert, Elisabeth Davioud-Charvet

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 129 KB

english, 2002

8

Structure–activity relationships of the peptide deformylase inhibitor BB-3497: modification of the metal binding group

Helen K. Smith, R.Paul Beckett, John M. Clements, Sheila Doel, Stephen P. East, Steven B. Launchbury, Lisa M. Pratt, Zoë M. Spavold, Wayne Thomas, Richard S. Todd, Mark Whittaker

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 161 KB

english, 2002

9

Synthesis and pharmacological evaluation of a new class of peroxisome proliferator-activated receptor modulators

Markus Thor, Katarina Beierlein, Graeme Dykes, Anna-Lena Gustavsson, Jessica Heidrich, Lena Jendeberg, Bengt Lindqvist, Cecile Pegurier, Patrick Roussel, Martin Slater, Stefan Svensson, Mona Sydow-Bäc

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 152 KB

english, 2002

10

A simple and rapid method for the differentiation of C-13 manoyl oxide epimers in biologically important samples using GC–MS analysis supported with NMR spectroscopy and computational chemistry results

Costas Demetzos, Antonios Kolocouris, Thalia Anastasaki

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 220 KB

english, 2002

11

Synthesis and biological evaluation of novel 2-(1H-imidazol-4-yl)cyclopropane carboxylic acids: key intermediates for H3 histamine receptor ligands

Miguel F Braña, Cristina Guisado, Luis Fernando Alguacil, Elisa Garrido, Carmen Pérez-Garcı́a, Mariano Ruiz-Gayo

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 124 KB

english, 2002

12

Synthesis and biological evaluation of aristolactams

Axel Couture, Eric Deniau, Pierre Grandclaudon, Hélène Rybalko-Rosen, Stéphane Léonce, Bruno Pfeiffer, Pierre Renard

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 126 KB

english, 2002

13

Nitrite-Mediated decarboxylative conjugation of caffeic acid with glutathione under mildly acidic conditions

Lucia Panzella, Alessandra Napolitano, Marco d'Ischia

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 114 KB

english, 2002

14

17S,20S-Methanofusidic acid, a new potent semi-synthetic fusidane antibiotic

Tore Duvold, Anne Jørgensen, Niels R. Andersen, Anne S. Henriksen, Morten Dahl Sørensen, Fredrik Björkling

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 171 KB

english, 2002

15

Natural and synthetic geiparvarins are strong and selective MAO-B inhibitors. synthesis and SAR studies

Angelo Carotti, Antonio Carrieri, Stefano Chimichi, Marco Boccalini, Barbara Cosimelli, Carmela Gnerre, Andrea Carotti, Pierre-Alain Carrupt, Bernard Testa

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 184 KB

english, 2002

16

Synthetic studies of cis-4-Amino-l-proline derivatives as novel lipid lowering agents

Saibal Kumar Das, V.L. Narasimha Rao Krovvidi, H. Jagadheshan, Javed Iqbal

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 132 KB

english, 2002

17

Synthesis of aglycon analogues of sarmentosin and Their bioactivity of lymphocyte proliferation

Hong Zhang, Rui Xu, Zhongliang Hu, Xuchang He, Donglu Bai, Xiaoyu Li, Xiaofeng Wang

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 110 KB

english, 2002

18

Silanediol-Based inhibitor of thermolysin

Jaeseung Kim, Athanasios Glekas, Scott McN Sieburth

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 132 KB

english, 2002

19

Stereoselective and improved syntheses and anticancer testing of 3′-O-silatranylthymidines

Christine A. Black, Jason W. Ucci, Jeremy S. Vorpagel, Matthew C. Mauck, Edward E. Fenlon

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 118 KB

english, 2002

20

Synthesis of (+)-Lasonolide A: (−)-Lasonolide A is the biologically active enantiomer

Eun Lee, Ho Young Song, Jung Min Joo, Jung Won Kang, Dae Shik Kim, Cheol Kyu Jung, Chang Yong Hong, ShinWu Jeong, Kiwan Jeon

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 107 KB

english, 2002

21

Synthesis and cytotoxic activity of a new potent daunomycinone derivative

Nectarios Aligiannis, Nicole Pouli, Panagiotis Marakos, Alexios-Leandros Skaltsounis, Harris Pratsinis

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 123 KB

english, 2002

22

Optimization of a pyrazolo[1,5-a]pyrimidine class of KDR kinase inhibitors: improvements in physical properties enhance cellular activity and pharmacokinetics

Mark E. Fraley, Robert S. Rubino, William F. Hoffman, Scott R. Hambaugh, Kenneth L. Arrington, Randall W. Hungate, Mark T. Bilodeau, Andrew J. Tebben, Ruth Z. Rutledge, Richard L. Kendall, Rosemary C.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 175 KB

english, 2002

23

Contributors to this Issue

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 42 KB

english, 2002

24

Graphical Abstracts

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 214 KB

english, 2002

25

Instructions to Contributors

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 103 KB

english, 2002

26

Author Index 2002

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

File:

PDF, 166 KB

2002

27

Volume Contents 2002

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 327 KB

english, 2002

28

Inhibition of amine oxidases activity by 1-acetyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole derivatives

Fedele Manna, Franco Chimenti, Adriana Bolasco, Daniela Secci, Bruna Bizzarri, Olivia Befani, Paola Turini, Bruno Mondovı̀, Stefano Alcaro, Andrea Tafi

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 202 KB

english, 2002

29

Scanning the prime-Site substrate specificity of proteolytic enzymes: A novel assay based on ligand-Enhanced lanthanide ion fluorescence

Amy M. Barrios, Charles S. Craik

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 231 KB

english, 2002

30

2-(Dimethylaminomethyl)-tetrahydroisoxazolopyridobenzazepine derivatives. Synthesis of a new 5-HT2C antagonist with potential anxiolytic properties

J.Ignacio Andrés, José M. Alonso, Javier Fernández, Laura Iturrino, Pedro Martı́nez, Theo F. Meert, Victor K. Sipido

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 156 KB

english, 2002

31

Design and efficient synthesis of new stable 1α,25-dihydroxy-19-norvitamin D3 analogues containing amide bond

Yoshitomo Suhara, Atsushi Kittaka, Keiichiro Ono, Masaaki Kurihara, Toshie Fujishima, Akihiro Yoshida, Hiroaki Takayama

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 194 KB

english, 2002

32

Isolation and antimalarial activity of peroxydisulfate oxidation products of primaquine

Virendra K Dua, Sukesh N Sinha, Sukla Biswas, N Valecha, S.K Puri, V.P Sharma

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 119 KB

english, 2002

33

Synthesis of new targretin® analogues that induce apoptosis in leukemia HL-60 cells

Jean-Yves Winum, Stephen Baghdiguian, Thérèse Commes, Alain Leydet, Jean-Louis Montero

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 265 KB

english, 2002

34

Erratum to “Tryptophanyl phosphoramidates as prodrugs of synadenol and its E-isomer: synthesis and biological activity” [Bioorg. Med. Chem. Lett. 12 (2002) 2467]

Ruifang Wang, Thomas H Corbett, Yung-Chi Cheng, John C Drach, Earl R Kern, Hiroaki Mitsuya, Jiri Zemlicka

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 64 KB

english, 2002

35

Vacuolar-type H+-ATPase inhibitory activity of synthetic analogues of the concanamycins: Is the hydrogen bond network involving the lactone carbonyl, the hemiacetal hydroxy group, and the C-19 hydroxy group essential for the biological activity of the concanamycins?

Yuya Yoshimoto, Takaaki Jyojima, Tsuyoshi Arita, Minoru Ueda, Masaya Imoto, Shuichi Matsumura, Kazunobu Toshima

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 183 KB

english, 2002

36

A novel synthesis of d-galactofuranosyl, d-glucofuranosyl and d-mannofuranosyl 1-phosphates based on remote activation of new and free hexofuranosyl donors

Vincent Ferrières, Sophie Blanchard, Delphine Fischer, Daniel Plusquellec

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 140 KB

english, 2002

37

Bioactive 4-substituted-6-methyl-2-pyrones with promising cytotoxicity against A2780 and K562 cell lines

Lester R. Marrison, Julia M. Dickinson, Ian J.S. Fairlamb

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 138 KB

english, 2002

38

Inside (Editorial Board)

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 53 KB

english, 2002

39

Contents List

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 113 KB

english, 2002

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