Volume 30; Issue 19

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Bioorganic & Medicinal Chemistry Letters
Volume 30; Issue 19

Bioorganic & Medicinal Chemistry Letters

Volume 30; Issue 19

1

2H-1,2,3-Triazole-chalcones as novel cytotoxic agents against prostate cancer

Pinheiro, Sergio, PessÃ´a, Jaqueline C., Pinheiro, Erick M.C., Muri, Estela M.F., Filho, Eclair Venturini, Loureiro, Laiza B., Freitas, Maria Clara R., Silva Junior, Carlos M.D., Fiorot, Rodolfo G., C

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 1.39 MB

2020

2

Discovery of novel (6S/12aS)-heptachpyridone capable of inhibiting thrombosis in vivo

Hou, Mengyu, Lv, Manjie, Zhang, Xiaoyi, Wang, Yaonan, Zhao, Shurui, Wu, Jianhui, Peng, Shiqi, Zhao, Ming

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 1.22 MB

2020

3

Synthesis and biological evaluation of ethacrynic acid derivatives bearing sulfonamides as potent anti-cancer agents

El Abbouchi, Abdelmoula, El Brahmi, Nabil, Hiebel, Marie-Aude, Bignon, JÃ©rÃ´me, Guillaumet, GÃ©rald, Suzenet, Franck, El Kazzouli, SaÃ¯d

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 416 KB

2020

4

Correlations between functional porphyrin positions and accumulation in cancer cells

Tojo, Toshifumi, Nishida, Koshi, Kondo, Takeshi, Yuasa, Makoto

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 1.81 MB

2020

5

Mechanistic insights into the activation of ester prodrugs of 666-15

Xie, Fuchun, MartÃn-Acosta, Pedro, Li, Bingbing X., Xiao, Xiangshu

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 1.38 MB

2020

6

Structure activity study of S-trityl-cysteamine dimethylaminopyridine derivatives as SIRT2 inhibitors: Improvement of SIRT2 binding and inhibition

Radwan, Mohamed O., Ciftci, Halil I., Ali, Taha F.S., Koga, Ryoko, Tateishi, Hiroshi, Nakata, Akiko, Ito, Akihiro, Yoshida, Minoru, Fujita, Mikako, Otsuka, Masami

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 1.74 MB

2020

7

Synthesis and biological effect of lysosome-targeting fluorescent anion transporters with enhanced anionophoric activity

Hong, Xiao-Qiao, He, Xiang-Yu, Tam, Kin Yip, Chen, Wen-Hua

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 1.87 MB

2020

8

Discovery of 2,6âdifluorobenzyl ether series of phenyl ((R)â3âphenylpyrrolidinâ3âyl)sulfones as surprisingly potent, selective and orally bioavailable RORÎ³t inverse agonists

Duan, James J.-W., Jiang, Bin, Lu, Zhonghui, Stachura, Sylwia, Weigelt, Carolyn A., Sack, John S., Khan, Javed, Ruzanov, Max, Wu, DauhâRurng, Yarde, Melissa, Shen, DingâRen, Zhao, Qihong, Salterâ

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 2.25 MB

2020

9

Annulation reaction enables the identification of an exocyclic amide tricyclic chemotype as retinoic acid Receptor-Related orphan receptor gamma (RORÎ³/RORc) inverse agonists

Marcoux, David, Bertrand, Myra Beaudoin, Weigelt, Carolyn A., Yip, Shiuhang, Galella, Michael, Park, Hyunsoo, Wu, Dauh-Rurng, Wang, Jinhong, Yarde, Melissa, Cvijic, Mary Ellen, Li, Sha, Hynes, John, T

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 734 KB

2020

10

Editorial Board

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 34 KB

2020

11

Graphical abstract TOC

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 148 KB

2020

12

Graphical abstract TOC

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 345 KB

2020

13

Graphical Abstract Contents Continued

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 263 KB

2020